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PreprintAll rights reservedbioRxiv

Discovery of a molecular glue inhibitor that stabilises a non-productive Kalirin-Rac1 complex

  • J. L. Gray
  • M. C. Callens
  • A. Henley
  • D. Zaidman
  • C. Jimenez Antunez
  • A. P. Thompson
  • Z. Lei
  • R. Skyner
  • M. Miller
  • E. P. Williams
  • A. Robinson
  • R. Seupal
7 more authors
  • M. T. Fry
  • M. Filep
  • F. von Delft
  • M. P. Willis
  • A. R. von Delft
  • N. London
  • P. E. Brennan1
  1. 1University of Oxford
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Cite

BibTeXRIS
BibTeX
@misc{gray2026discovery,
  title = {{Discovery of a molecular glue inhibitor that stabilises a non-productive Kalirin-Rac1 complex}},
  author = {J. L. Gray and M. C. Callens and A. Henley and D. Zaidman and C. Jimenez Antunez and A. P. Thompson and Z. Lei and R. Skyner and M. Miller and E. P. Williams and A. Robinson and R. Seupal and M. T. Fry and M. Filep and F. von Delft and M. P. Willis and A. R. von Delft and N. London and P. E. Brennan},
  howpublished = {bioRxiv},
  year = {2026},
  month = sep,
  doi = {10.64898/2026.09.08.749156},
  url = {https://www.biorxiv.org/content/10.64898/2026.09.08.749156v1},
}
RIS
TY  - UNPB
TI  - Discovery of a molecular glue inhibitor that stabilises a non-productive Kalirin-Rac1 complex
AU  - J. L. Gray
AU  - M. C. Callens
AU  - A. Henley
AU  - D. Zaidman
AU  - C. Jimenez Antunez
AU  - A. P. Thompson
AU  - Z. Lei
AU  - R. Skyner
AU  - M. Miller
AU  - E. P. Williams
AU  - A. Robinson
AU  - R. Seupal
AU  - M. T. Fry
AU  - M. Filep
AU  - F. von Delft
AU  - M. P. Willis
AU  - A. R. von Delft
AU  - N. London
AU  - P. E. Brennan
PY  - 2026
DA  - 2026/09/08
PB  - bioRxiv
DO  - 10.64898/2026.09.08.749156
UR  - https://www.biorxiv.org/content/10.64898/2026.09.08.749156v1
ER  -