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Peer-reviewedPublisher termsRSC Medicinal Chemistry

DprE1 inhibitors in tuberculosis: integrating structural binding determinants, IC50–MIC translation, and physicochemical constraints for rational drug design

  • Fady H. Fayek1
  • Mai H. A. Mousa1
  • Mona F. Said2
  • Hanan H. Georgey1,2
  • Nagwa M. Abdel Gawad2
  1. 1Department of Pharmaceutical Chemistry, Faculty of Pharmacy and Drug Technology, Egyptian Chinese University Gesr El Suez street, PO 11786 Cairo Egypt
  2. 2Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Cairo University Kasr El-Aini Street, P.O. Box 11562 Cairo Egypt
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Cite

BibTeXRIS
BibTeX
@article{fayek2026dpre1,
  title = {{DprE1 inhibitors in tuberculosis: integrating structural binding determinants, IC50–MIC translation, and physicochemical constraints for rational drug design}},
  author = {Fady H. Fayek and Mai H. A. Mousa and Mona F. Said and Hanan H. Georgey and Nagwa M. Abdel Gawad},
  journal = {RSC Medicinal Chemistry},
  year = {2026},
  month = nov,
  doi = {10.1039/d6md00729e},
  url = {https://doi.org/10.1039/d6md00729e},
}
RIS
TY  - JOUR
TI  - DprE1 inhibitors in tuberculosis: integrating structural binding determinants, IC50–MIC translation, and physicochemical constraints for rational drug design
AU  - Fady H. Fayek
AU  - Mai H. A. Mousa
AU  - Mona F. Said
AU  - Hanan H. Georgey
AU  - Nagwa M. Abdel Gawad
PY  - 2026
DA  - 2026/11/04
JO  - RSC Medicinal Chemistry
DO  - 10.1039/d6md00729e
UR  - https://doi.org/10.1039/d6md00729e
SN  - 2632-8682
ER  -