Peer-reviewedLicence not statedBioorganic and Medicinal Chemistry Letters
Synthesis and radioligand binding studies of bis-(8-isopropyl-isoquinolinium) derivatives as ligands for apamin-sensitive sites on cloned SK2 and SK3 channels
Related
- Fragment‐Linked Purine Derivatives as Inhibitors of (p)ppGpp Synthetases: Design, Synthesis, and Structure‐Activity Relationships
- Synthesis of 1,2,3-Triazole Derivatives of N,N-Dimethyltryptamine Isolated From Mimosa tenuiflora Root Bark: Antiplasmodial Activity In Silico and In Vitro.
- Novel Quinoxaline-Based Cyanocarbonimidodithioate Derivatives as Non-Hydroxamate Selective HDAC8 Inhibitors: Design, Synthesis, Biological Evaluation and Mechanistic Studies
- Design, Synthesis, Evaluation, and Molecular Dynamics Simulation of Tadalafil Derivatives for the Treatment of Erectile Dysfunction
- Design, synthesis, and evaluation of novel hydrazide and hydroxamate derivatives as potent antileukemic agents with preferential HDAC-2 inhibitory activity over class I isoform
BibTeX
@article{badarau2026synthesis,
title = {{Synthesis and radioligand binding studies of bis-(8-isopropyl-isoquinolinium) derivatives as ligands for apamin-sensitive sites on cloned SK2 and SK3 channels}},
author = {Eduard Badarau and Sébastien Dilly and Fabien Dufour and Sylvie Poncin and Vincent Seutin and Jean-François Liégeois},
journal = {Bioorganic and Medicinal Chemistry Letters},
year = {2026},
month = oct,
doi = {10.1016/j.bmcl.2011.09.043},
url = {https://hal.science/hal-05793324v1},
}
RIS
TY - JOUR
TI - Synthesis and radioligand binding studies of bis-(8-isopropyl-isoquinolinium) derivatives as ligands for apamin-sensitive sites on cloned SK2 and SK3 channels
AU - Eduard Badarau
AU - Sébastien Dilly
AU - Fabien Dufour
AU - Sylvie Poncin
AU - Vincent Seutin
AU - Jean-François Liégeois
PY - 2026
DA - 2026/10/12
JO - Bioorganic and Medicinal Chemistry Letters
DO - 10.1016/j.bmcl.2011.09.043
UR - https://hal.science/hal-05793324v1
SN - 0960-894X
ER -