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Peer-reviewedPublisher termsRSC Medicinal Chemistry

Discovery of an NRAS isoform and activation-state selective macrocyclic peptide

  • Kenneth K. Hallenbeck1
  • Yunpeng Zhou1
  • Hubert Josien2
  • Songnian Lin2
  • Aileen Soriano1
  • Todd Mayhood1
  • Jaclyn Robustelli1
  • Xiaomei Chai1
  • My Sam Mansueto1
  • Gireedhar Venkatachalam3
  • Ryan E. Loy1
  • Erwin G. Abucayon4
7 more authors
  • Peng-Hsun Chase Chen1
  • Huifang Yao1
  • Haihong Zhou1
  • Elsa B. Krall5
  • David G. McLaren1
  • Adam Weinglass1
  • S. Adrian Saldanha1
5 affiliations
  1. 1Quantitative Biosciences, Merck & Co., Inc. Rahway NJ 07065 USA
  2. 2Discovery Chemistry, Merck & Co., Inc. Rahway NJ 07065 USA
  3. 3Quantitative Biosciences, MSD International Singapore
  4. 4Analytical Research & Development, Merck & Co., Inc. Rahway NJ 07065 USA
  5. 5Discovery Oncology, Merck & Co., Inc. Rahway NJ 07065 USA
Read full textDOICite

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Cite

BibTeXRIS
BibTeX
@article{hallenbeck2026discovery,
  title = {{Discovery of an NRAS isoform and activation-state selective macrocyclic peptide}},
  author = {Kenneth K. Hallenbeck and Yunpeng Zhou and Hubert Josien and Songnian Lin and Aileen Soriano and Todd Mayhood and Jaclyn Robustelli and Xiaomei Chai and My Sam Mansueto and Gireedhar Venkatachalam and Ryan E. Loy and Erwin G. Abucayon and Peng-Hsun Chase Chen and Huifang Yao and Haihong Zhou and Elsa B. Krall and David G. McLaren and Adam Weinglass and S. Adrian Saldanha},
  journal = {RSC Medicinal Chemistry},
  year = {2026},
  month = oct,
  doi = {10.1039/d6md00720a},
  url = {https://doi.org/10.1039/d6md00720a},
}
RIS
TY  - JOUR
TI  - Discovery of an NRAS isoform and activation-state selective macrocyclic peptide
AU  - Kenneth K. Hallenbeck
AU  - Yunpeng Zhou
AU  - Hubert Josien
AU  - Songnian Lin
AU  - Aileen Soriano
AU  - Todd Mayhood
AU  - Jaclyn Robustelli
AU  - Xiaomei Chai
AU  - My Sam Mansueto
AU  - Gireedhar Venkatachalam
AU  - Ryan E. Loy
AU  - Erwin G. Abucayon
AU  - Peng-Hsun Chase Chen
AU  - Huifang Yao
AU  - Haihong Zhou
AU  - Elsa B. Krall
AU  - David G. McLaren
AU  - Adam Weinglass
AU  - S. Adrian Saldanha
PY  - 2026
DA  - 2026/10/22
JO  - RSC Medicinal Chemistry
DO  - 10.1039/d6md00720a
UR  - https://doi.org/10.1039/d6md00720a
SN  - 2632-8682
ER  -