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Peer-reviewedPublisher termsEuropean Journal of Medicinal Chemistry

Fragment-based drug discovery strategy reveals an unprecedented allosteric binding site in Mycobacterium tuberculosis DNA gyrase

  • Sabrina Tami Shiroma
  • Nicolas de Oliveira Rossini
  • Jillian F Armenia
  • Catharina dos Santos Silva
  • Paulo C.T. Souza
  • Pierre-Damien Coureux
  • Neil Osheroff
  • Marcio V.B. Dias
Open at sourcePDFDOICite

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Cite

BibTeXRIS
BibTeX
@article{shiroma2026fragmentbased,
  title = {{Fragment-based drug discovery strategy reveals an unprecedented allosteric binding site in Mycobacterium tuberculosis DNA gyrase}},
  author = {Sabrina Tami Shiroma and Nicolas de Oliveira Rossini and Jillian F Armenia and Catharina dos Santos Silva and Paulo C.T. Souza and Pierre-Damien Coureux and Neil Osheroff and Marcio V.B. Dias},
  journal = {European Journal of Medicinal Chemistry},
  year = {2026},
  month = sep,
  doi = {10.1016/j.ejmech.2026.119380},
  url = {https://hal.science/hal-05787654v1},
}
RIS
TY  - JOUR
TI  - Fragment-based drug discovery strategy reveals an unprecedented allosteric binding site in Mycobacterium tuberculosis DNA gyrase
AU  - Sabrina Tami Shiroma
AU  - Nicolas de Oliveira Rossini
AU  - Jillian F Armenia
AU  - Catharina dos Santos Silva
AU  - Paulo C.T. Souza
AU  - Pierre-Damien Coureux
AU  - Neil Osheroff
AU  - Marcio V.B. Dias
PY  - 2026
DA  - 2026/09/29
JO  - European Journal of Medicinal Chemistry
DO  - 10.1016/j.ejmech.2026.119380
UR  - https://hal.science/hal-05787654v1
SN  - 0223-5234
SN  - 1768-3254
ER  -